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drug receptor binding

"Synthesis of new C-25 and C-26 steroidal acids as potential ligands of the nuclear receptors DAF-12, LXR and GR" (2017) Dansey, M.V.; del Fueyo, M.C.; Veleiro, A.S.; Di Chenna, P.H. Steroids. 121:40-46

"Synthetic stigmastanes with dual antiherpetic and immunomodulating activities inhibit ERK and Akt signaling pathways without binding to glucocorticoid receptors" (2016) Michelini, F.M.;Bueno, C.A.;Molinari, A.M. (...)Ramírez, J.A. Biochimica et Biophysica Acta - General Subjects. 1860(1):129-139

"The estrogen receptor alpha nuclear localization sequence is critical for fulvestrant-induced degradation of the receptor" (2015) Casa, A.J.;Hochbaum, D.;Sreekumar, S. (...)Lee, A.V. Molecular and Cellular Endocrinology. 415:76-86

"Effect of synthetic steroids on GABAA receptor binding in rat brain" (2015) Rey, M.;Veleiro, A.S.;Ghini, A.A. (...)Coirini, H. Neuroscience. 290:138-146

"The selective glucocorticoid receptor modulator CORT108297 restores faulty hippocampal parameters in Wobbler and corticosterone-treated mice" (2014) Meyer, M.;Gonzalez Deniselle, M.C.;Hunt, H. (...)De Nicola, A.F. Journal of Steroid Biochemistry and Molecular Biology. 143:40-48

"27-Nor-Δ4-dafachronic acid is a synthetic ligand of Caenorhabditis elegans DAF-12 receptor" (2013) Samaja, G.A.;Castro, O.;Alvarez, L.D. (...)Burton, G. Bioorganic and Medicinal Chemistry Letters. 23(10):2893-2896

"Neuroprotective action of synthetic steroids with oxygen bridge. Activity on GABAA receptor" (2013) Rey, M.;Kruse, M.S.;Alvarez, L.D. (...)Coirini, H. Experimental Neurology. 249:49-58

"Effect of SOM230 (Pasireotide) on corticotropic cells: Action in dogs with Cushing's disease" (2011) Castillo, V.;Theodoropoulou, M.;Stalla, J. (...)Arzt, E. Neuroendocrinology. 94(2):124-136

"Structure of the glucocorticoid receptor, a flexible protein that can adapt to different ligands" (2010) Veleiro, A.S.; Alvarez, L.D.; Eduardo, S.L.; Burton, G. ChemMedChem. 5(5):649-659

"Insights on glucocorticoid receptor activity modulation through the binding of rigid steroids" (2010) Presman, D.M.;Alvarez, L.D.;Levi, V. (...)Pecci, A. PLoS ONE. 5(10)

"New lead compounds in the search for pure antiglucocorticoids and the dissociation of antiglucocorticoid effects" (2009) Pecci, A.;Alvarez, L.D.;Veleiro, A.S. (...)Burton, G. Journal of Steroid Biochemistry and Molecular Biology. 113(3-5):155-162

"Structure-activity relationships of neuroactive steroids acting on the GABAA receptor" (2009) Veleiro, A.S.; Burton, G. Current Medicinal Chemistry. 16(4):455-472

"Synthesis and GABAA receptor activity of 2,19-sulfamoyl analogues of allopregnanolone" (2009) Durán, F.J.;Edelsztein, V.C.;Ghini, A.A. (...)Burton, G. Bioorganic and Medicinal Chemistry. 17(18):6526-6533

"Alpha9 nicotinic acetylcholine receptors and the treatment of pain" (2009) McIntosh, J.M.;Absalom, N.;Chebib, M. (...)Vincler, M. Biochemical Pharmacology. 78(7):693-702

"Synthesis and GABAA receptor activity of oxygen-bridged neurosteroid analogs" (2008) Alvarez, L.D.;Veleiro, A.S.;Baggio, R.F. (...)Burton, G. Bioorganic and Medicinal Chemistry. 16(7):3831-3838

"Synthesis of 6-thia analogs of the natural neurosteroid allopregnanolone" (2006) Durán, F.J.; Ghini, A.A.; Coirini, H.; Burton, G. Tetrahedron. 62(20):4762-4768

"Heparin increases the adhesion of murine mammary adenocarcinoma cells (LM3). Correlation with the presence of heparin receptors on cell surface" (2005) Bertolesi, G.; Eijan, A.M.; Calvo, J.C.; de Cidre, L.L. Journal of Biological Regulators and Homeostatic Agents. 19(1-2):33-40

"Effects of quinine, quinidine, and chloroquine on α9α10 nicotinic cholinergic receptors" (2005) Ballestero, J.A.;Plazas, P.V.;Kracun, S. (...)Elgoyhen, A.B. Molecular Pharmacology. 68(3):822-829

"Studies on the mechanisms of action of picrotoxin, quercetin and pregnanolone at the GABA ρ1 receptor" (2004) Goutman, J.D.; Calvo, D.J. British Journal of Pharmacology. 141(4):717-727

"Tiotidine, a histamine H2 receptor inverse agonist that binds with high affinity to an inactive G-protein-coupled form of the receptor. Experimental support for the cubic ternary complex model" (2003) Monczor, F.;Fernández, N.;Legnazzi, B.L. (...)Davio, C. Molecular Pharmacology. 64(2):512-520

"Direct interaction of serotonin type 3 receptor ligands with recombinant and native α9α10-containing nicotinic cholinergic receptors" (2003) Rothlin, C.V.;Lioudyno, M.I.;Silbering, A.F. (...)Elgoyhen, A.B. Molecular Pharmacology. 63(5):1067-1074

"Functional expression and properties of a nicotinic α9/5-HT3 A chimeric receptor" (2003) Verbitsky, M.; Plazas, P.V.; Elgoyhen, A.B. NeuroReport. 14(15):1931-1934

"Cocaine-induced locomotor activity and cocaine discrimination in dopamine D2 receptor mutant mice" (2002) Chausmer, A.L.;Elmer, G.I.;Rubinstein, M. (...)Katz, J.L. Psychopharmacology. 163(1):54-61

"Molecular modelling of the interactions of carbamazepine and a nicotinic receptor involved in the autosomal dominant nocturnal frontal lobe epilepsy" (2002) Ortells, M.O.; Barrantes, G.E. British Journal of Pharmacology. 136(6):883-895

"Correlation between pregnanesteroid conformation, receptor affinity, and anti-natriuretic effect" (2002) Piwien-Pilipuk, G.; Kanelakis, K.C.; Galigniana, M.D. European Journal of Pharmacology. 454(2-3):131-143

"Androgen receptors in human melanoma cell lines IIB-MEL-LES and IIB-MEL-IAN and in human melanoma metastases" (2002) Morvillo, V.;Lüthy, I.A.;Bravo, A.I. (...)Mordoh, J. Melanoma Research. 12(6):529-538

"Dopamine D4 receptor-deficient mice display cortical hyperexcitability" (2001) Rubinstein, M.;Cepeda, C.;Hurst, R.S. (...)Grandy, D.K. Journal of Neuroscience. 21(11):3756-3763

"An astroglia-linked dopamine D2-receptor action in prefrontal cortex" (2001) Khan, Z.U.;Koulen, P.;Rubinstein, M. (...)Goldman-Rakic, P.S. Proceedings of the National Academy of Sciences of the United States of America. 98(4):1964-1969

"α10: A determinant of nicotinic cholinergic receptor function in mammalian vestibular and cochlear mechanosensory hair cells" (2001) Elgoyhen, A.B.;Vetter, D.E.;Katz, E. (...)Boulter, J. Proceedings of the National Academy of Sciences of the United States of America. 98(6):3501-3506

"6-Chloro-3'-nitroflavone is a potent ligand for the benzodiazepine binding site of the GABA(A) receptor devoid of intrinsic activity" (2000) Viola, H.;Wolfman, C.;Marder, M. (...)Medina, J.H. Pharmacology Biochemistry and Behavior. 65(2):313-320

"Mixed nicotinic-muscarinic properties of the α9 nicotinic cholinergic receptor" (2000) Verbitsky, M.; Rothlin, C.V.; Katz, E.; Belén Elgoyhen, A. Neuropharmacology. 39(13):2515-2524

"Block of the α9 nicotinic receptor by ototoxic aminoglycosides" (2000) Rothlin, C.V.;Katz, E.;Verbitsky, M. (...)Elgoyhen, A.B. Neuropharmacology. 39(13):2525-2532

"Acyclic analogues of deoxyadenosine 3',5'-bisphosphates as P2Y 1 receptor antagonists" (2000) Kim, Y.-C.;Gallo-Rodriguez, C.;Jang, S.-Y. (...)Jacobson, K.A. Journal of Medicinal Chemistry. 43(4):746-755

"Mechanism of action of the potent sodium-retaining steroid 11,19- oxidoprogesterone" (2000) Galigniana, M.D.;Vicent, G.P.;Piwien-Pilipuk, G. (...)Lantos, C.P. Molecular Pharmacology. 58(1):58-70

"Angiotensin II-induced Ca2+ mobilization and prolactin release in normal and hyperplastic pituitary cells" (1998) Díaz-Torga, G.;Iglesias, A.G.;Achával-Zaia, R. (...)Becú-Villalobos, D. American Journal of Physiology - Endocrinology and Metabolism. 274(3 37-3):E534-E540

"Differential modulation of dopamine D 1 -receptor binding and mRNA expression in the basal ganglia by the D 1 -receptor antagonist, SCH-23390" (1998) Yu, J.;Coirini, H.;Källström, L. (...)Johnson, A.E. Synapse. 30(1):38-48

"21-hydroxy-6,19-oxidoprogesterone: A novel synthetic steroid with specific antiglucocorticoid properties in the rat" (1997) Vicent, G.P.;Monteserín, M.C.;Veleiro, A.S. (...)Galigniana, M.D. Molecular Pharmacology. 52(4):749-753

"Voltage-dependent calcium channels and G(i) regulatory protein mediate the human sperm acrosomal exocytosis induced by N-acetylglucosaminyl/mannosyl neoglycoproteins" (1996) Brandelli, A.; Miranda, P.V.; Tezón, J.G. Journal of Andrology. 17(5):522-529

"Binding of the anti-inflammatory steroid deflazacort to glucocorticoid receptors in brain and peripheral tissues. In vivo and in vitro studies" (1994) Coirini, H.;Flores, D.;Cristina Vega, M. (...)De Nicola, A.F. Journal of Steroid Biochemistry and Molecular Biology. 49(1):43-49

"Effects of dopamine and tamoxifen on serum prolactin and nuclear estrogen receptors in rat anterior pituitaries" (1993) Stalldecker, G.;Reynoso, R.;Piroli, G. (...)De Nicola, A.F. Neuroendocrinology Letters. 15(5-6):389-395

"Physiological, biochemical and molecular mechanisms of salt appetite control by mineralocorticoid action in brain" (1992) De Nicola, A.F.; Grillo, C.; Gonzalez, S. Brazilian Journal of Medical and Biological Research. 25(12):1153-1162

"Glucocorticoid type II receptors of the spinal cord show lower affinity than hippocampal type II receptors: Binding parameters obtained with different experimental protocols" (1991) Moses, D.F.; González, S.; McEwen, B.S.; De Nicola, A.F. Journal of Steroid Biochemistry and Molecular Biology. 39(1):5-12

"Role of thromboxanes in alterations of the diabetic β-adrenergic system" (1989) Wald, M.; Pascual, J.; Sterin-Borda, L. Biochemical Pharmacology. 38(19):3347-3355

"Uptake and release of 3H prostaglandins E2 and F2α in uterin strips isolated from ovariectomized rats. Influence of in vitro progesterone" (1987) Gimeno, M.F.; Franchi, A.M.; González, E.T.; Gimeno, A.L. Prostaglandins. 33(1):51-61

"Changes in gamma-aminobutyric acid high affinity binding to cerebral cortex membranes after pinealectomy or melatonin administration to rats1" (1986) Castroviejo, D.A.; Rosenstein, R.E.; Romeo, H.E.; Cardinali, D.P. Neuroendocrinology. 43(1):24-31

"Binding and effects of catecholestrogens on adenylate cyclase activity, and adrenoceptors, benzodiazepine and GABA receptors in guinea-pig hypothalamic membranes" (1986) Etchegoyen, G.S.;Cardinali, D.P.;Pérez, A.E. (...)Pérez-Palacios, G. European Journal of Pharmacology. 129(1-2):1-10

"Role of β2-adrenoceptors in the biological effect of autoimmune orchitis spleen cells" (1986) Borda, E.; Perez Leiros, C.; Sterin-Borda, L. Canadian Journal of Physiology and Pharmacology. 64(8):1091-1095

"Diurnal Variations of Benzodiazepine Binding in Rat Cerebral Cortex: Disruption by Pinealectomy" (1986) Acuña‐Castroviejo, D.; Lowenstein, P.R.; Rosenstein, R.; Cardinali, D.P. Journal of Pineal Research. 3(2):101-109

"Melatonin increases in vivo GABA accumulation in rat hypothalamus, cerebellum, cerebral cortex and pineal gland" (1986) Rosenstein, R.E.; Cardinali, D.P. Brain Research. 398(2):403-406

"Effect of androgen on androgen receptors in cultured human epididymis" (1986) Vazquez, M.H.; De Larminat, M.A.; Blaquier, J.A. Journal of Endocrinology. 111(2):343-348

"ᵦ-(-4 Chlorophenyl) GABA (Baclofen) Inhibits Prolactin and Thyrotropin Release by Acting on the Rat Brain" (1986) Lux, V.A.R.; Somoza, G.M.; Libertun, C. Proceedings of the Society for Experimental Biology and Medicine. 183(3):358-362

"Hormonal effects on unoccupied estrogen receptors in nuclei of anterior pituitary glands" (1986) Weisenberg, L.S.;Orti, E.;Piroli, G. (...)De Nicola, A.F. Acta Physiologica et Pharmacologica Latinoamericana. 36(4):473-487

"Bromocriptine and sulpiride competitively inhibit estrogen binding to its receptor in the adrenal gland" (1986) Lüthy, I.A.; Calandra, R.S. Experientia. 42(2):136-138

"Ontogenesis of [3H]serotonin binding sites in the hypothalamus of the female rat: Relation to serotonin-induced LH release in moxestrol-pretreated rats" (1986) Becú-Villalobos, D.; Libertun, C. Developmental Brain Research. 25(1):111-116

"Regulatory factors of glucocorticoid binding in early and term rat placenta" (1986) Heller, C.L.; Ortí, E.; De Nicola, A.F. Journal of Steroid Biochemistry. 25(1):53-58

"Alterations in the prolactin secretion in streptozotocin-induced diabetic rats. Correlation with pituitary and hypothalamus estradiol receptors" (1985) Tesone, M.; Ladenheim, R.G.; Charreau, E.H. Molecular and Cellular Endocrinology. 43(2-3):135-140

"Estradiol binding and phosphatase activity in the uterus after castration and chronic diabetes: Effect of molybdate and estrogen replacement" (1985) Fridman, O.; Moses, D.; De Nicola, A.F. Acta Physiologica et Pharmacologica Latinoamericana. 35(2):193-203

"Melatonin reverses pinealectomy-induced decrease of benzodiazepine binding in rat cerebral cortex" (1985) Lowenstein, P.R.; Rosenstein, R.; Cardinali, D.P. Neurochemistry International. 7(4):675-681

"Effects of the methylxanthine derivative pentoxifylline on benzodiazepine and muscarinic binding sites in rat cerebral cortex" (1985) Lowenstein, P.R.; Aguilar, J.S.O.; Sabato, U.C. Acta Physiologica et Pharmacologica Latinoamericana. 35(4):431-439

"Prolactin binding sites in the brain and kidneys of the toad, Bufo arenarum Hensel" (1985) Lüthy, I.A.;Segura, E.T.;Lüthy, V.I. (...)Calandra, R.S. Journal of Comparative Physiology B. 155(5):611-614

"Properties and distribution of glucocorticoid-binding sites in cytosol of the spinal cord" (1985) Orti, E.; Coirini, H.; De Nicola, A.F. Neuroendocrinology. 40(3):225-231

"Effect of median eminence lesions and hormonal replacement on the prolactin receptors in the adrenal Gland and langerhans islets from ovariectomized adult rats" (1985) Lüthy, I.A.;Tesone, M.;Oliveira-Filho, R.M. (...)Calandra, R.S. Journal of Receptors and Signal Transduction. 5(1):105-119

"In Vitro Uptake of Benzodiazepines by Rat Pineal Gland" (1984) Lowenstein, P.R.; Solveyra, C.G.; Cardinali, D.P. Journal of Pineal Research. 1(3):207-213

"Benzodiazepine binding sites in human pineal gland" (1984) Lowenstein, P.R.; Rosenstein, R.; Caputti, E.; Cardinali, D.P. European Journal of Pharmacology. 106(2):399-403

"Effects of prolactin, bromocriptine and sulpiride on estrogen and lactogenic receptors in the rat adrenal gland" (1984) Luthy, I.A.; Chiauzzi, V.A.; Charreau, E.H.; Calandra, R.S. Acta Physiologica et Pharmacologica Latinoamericana. 34(1):15-23

"Effect of a second injection of human chorionic gonadotropin on the desensitized Leydig cells" (1984) Calvo, J.C.; Radicella, J.P.; Pignataro, O.P.; Charreau, E.H. Molecular and Cellular Endocrinology. 34(1):31-38

"Insulin action and characterization of insulin receptors in rat luteal cells" (1984) Ladenheim, R.G.; Tesone, M.; Charreau, E.H. Endocrinology. 115(2):752-756

"A developmental study of adenohypophyseal dopaminergic receptors and of haloperidol-induced prolactin release in rats" (1984) Becúde Villalobos, D.; Vacas, M.I.; Cardinali, D.P.; Libertun, C. Developmental Brain Research. 12(2):167-171

"Prolactin regulation of prolactin binding sites in pancreatic islets and adrenal glands of ovariectomized rats" (1983) Tesone, M.; Luthy, I.A.; Ladenheim, R.G. Journal of Receptors and Signal Transduction. 3(6):711-726

"Androgens control androgen-binding sites in rat epididymis" (1983) Tezon, J.G.; Blaquier, J.A. Endocrinology. 113(3):1025-1030

"The placenta as a glucocorticoid target tissue: Exchange assay of (3H)-dexamethasone binding and effect of steroids on receptor content" (1983) Heller, C.; Coirini, H.; De Nicola, A.F. Hormone and Metabolic Research. 15(1):41-45

"Characterization of flunitrazepam and beta-carboline high affinity binding in bovine pineal gland" (1983) Lowenstein, P.R.; Cardinali, D.P. Neuroendocrinology. 37(2):150-154

"Hormone effects on muscarinic cholinergic binding in bovine and rat sympathetic superior cervical ganglia" (1983) Gejman, P.V.; Cardinali, D.P. Life Sciences. 32(9):965-972

"Benzodiazepine receptor sites in bovine pineal" (1982) Lowenstein, P.R.; Cardinali, D.P. European Journal of Pharmacology. 86(2):287-289

"Androgen determined subcellular distribution of receptor in rat epididymis" (1982) Tezon, J.G.; Vazquez, M.H.; Blaquier, J.A. Journal of Steroid Biochemistry. 17(3)