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Inhibitors
14
"Synthesis, molecular docking and biological evaluation of novel phthaloyl derivatives of 3-amino-3-aryl propionic acids as inhibitors of Trypanosoma cruzi trans-sialidase" (2018) Kashif, M.;Chacón-Vargas, K.F.;López-Cedillo, J.C. (...)Rivera, G. European Journal of Medicinal Chemistry. 156:252-268
"Thiodisaccharide sulfoxides: Absolute configuration of the so sulfur atom and influence on the biological activity towards the β-galactosidase from E. coli" (2015) Colomer, J.P.;Mayordomo, M.Á.C.;De Toro, B.F. (...)Varela, O. European Journal of Organic Chemistry. 2015(7):1448-1455
"Thiodisaccharide Sulfoxides: Absolute Configuration of the SO Sulfur Atom and Influence on the Biological Activity towards the β-Galactosidase from E. coli" (2015) Colomer, J.P.;Canales Mayordomo, M.A.;Fernández de Toro, B. (...)Varela, O. European Journal of Organic Chemistry
"Aryloxyethyl thiocyanates are potent growth inhibitors of Trypanosoma cruzi and Toxoplasma gondii" (2015) Chao, M.N.;Matiuzzi, C.E.;Storey, M. (...)Rodriguez, J.B. ChemMedChem. 10(6):1094-1108
"Improved bioavailability of inhibitors of Trypanosoma cruzi trans-sialidase: PEGylation of lactose analogs with multiarm polyethyleneglycol" (2012) Giorgi, M.E.;Ratier, L.;Agusti, R. (...)De Lederkremer, R.M. Glycobiology. 22(10):1363-1373
"Synthesis of oseltamivir conjugates with lactose analogs for inhibition studies on Trypanosoma cruzi trans-sialidase" (2011) Giorgi, M.E.; Piuselli, D.; Agusti, R.; De Lederkremer, R.M. Arkivoc. 2011(7):260-271
"Continuous nonradioactive method for screening trypanosomal transsialidase activity and its inhibitors" (2010) Sartor, P.A.;Agusti, R.;Leguizamón, M.S. (...)de Lederkremer, R.M. Glycobiology. 20(8):982-990
"Synthesis of PEGylated lactose analogs for inhibition studies on T.cruzi trans-sialidase" (2010) Giorgi, M.E.;Ratier, L.;Agusti, R. (...)De Lederkremer, R.M. Glycoconjugate Journal. 27(5):549-559
"Substrate stereo-specificity in tryptophan dioxygenase and indoleamine 2,3-dioxygenase" (2010) Capece, L.;Arrar, M.;Roitberg, A.E. (...)Estrin, D.A. Proteins: Structure, Function and Bioinformatics. 78(14):2961-2972
"Synthesis and evaluation of 1,1′-hydrocarbylenebis(indazol-3-ols) as potential antimalarial drugs" (2009) Alho, M.M.;García-Sánchez, R.N.;Nogal-Ruiz, J.J. (...)Arán, V.J. ChemMedChem. 4(1):78-87
"Lactose derivatives are inhibitors of Trypanosoma cruzi trans-sialidase activity toward conventional substrates in vitro and in vivo" (2004) Agustí, R.;París, G.;Ratier, L. (...)de Lederkremer, R.M. Glycobiology. 14(7):659-670
"Influence of exo β-D-galactofuranosidase inhibitors in cultures of Penicillium fellutanum and modifications in hyphal cell structure" (2002) Mariño, K.;Lima, C.;Maldonado, S. (...)De Lederkremer, R.M. Carbohydrate Research. 337(10):891-897