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Abstract:

We have described a method for preparation of [10B]-enriched-8- dihydroxyborylharmine (III) and characterized it by their spectral properties (MS, IR and NMR). This compound is a potential BNCT agent.

Registro:

Documento: Artículo
Título:A facile high-yield synthesis of [10B]-8-dihydroxyboryl harmine, a potential agent for boron neutron capture therapy
Autor:Sintas, J.A.; Macareno, N.J.; Vitale, A.A.
Filiación:Departamento de Quimica Organica, Fac. de Ciencias Exactas y Naturales, Universidad de Buenos Aires, 1428 Buenos Aires, Argentina
Palabras clave:8 dihydroxyborylharmine b 10; radiopharmaceutical agent; unclassified drug; animal tissue; autoradiography; binding site; conference paper; drug distribution; drug structure; drug synthesis; neutron capture therapy; nonhuman; rat
Año:2000
Volumen:5
Número:3
Página de inicio:526
Página de fin:528
DOI: http://dx.doi.org/10.3390/50300526
Título revista:Molecules
Título revista abreviado:Molecules
ISSN:14203049
CODEN:MOLEF
PDF:https://bibliotecadigital.exactas.uba.ar/download/paper/paper_14203049_v5_n3_p526_Sintas.pdf
Registro:https://bibliotecadigital.exactas.uba.ar/collection/paper/document/paper_14203049_v5_n3_p526_Sintas

Referencias:

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Citas:

---------- APA ----------
Sintas, J.A., Macareno, N.J. & Vitale, A.A. (2000) . A facile high-yield synthesis of [10B]-8-dihydroxyboryl harmine, a potential agent for boron neutron capture therapy. Molecules, 5(3), 526-528.
http://dx.doi.org/10.3390/50300526
---------- CHICAGO ----------
Sintas, J.A., Macareno, N.J., Vitale, A.A. "A facile high-yield synthesis of [10B]-8-dihydroxyboryl harmine, a potential agent for boron neutron capture therapy" . Molecules 5, no. 3 (2000) : 526-528.
http://dx.doi.org/10.3390/50300526
---------- MLA ----------
Sintas, J.A., Macareno, N.J., Vitale, A.A. "A facile high-yield synthesis of [10B]-8-dihydroxyboryl harmine, a potential agent for boron neutron capture therapy" . Molecules, vol. 5, no. 3, 2000, pp. 526-528.
http://dx.doi.org/10.3390/50300526
---------- VANCOUVER ----------
Sintas, J.A., Macareno, N.J., Vitale, A.A. A facile high-yield synthesis of [10B]-8-dihydroxyboryl harmine, a potential agent for boron neutron capture therapy. Molecules. 2000;5(3):526-528.
http://dx.doi.org/10.3390/50300526