Artículo
Rodriguez, J.B.; Zhong, L.; Docampo, R.; Wimmer, Z.; Gros, E.G. "Growth inhibitory effect of juvenile hormone analogues on epimastigotes of Trypanosoma cruzi" (1998) Bioorganic and Medicinal Chemistry Letters. 8(22):3257-3260
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Abstract:
Several compounds, structurally related to the insect growth regulator Fenoxycarb, exhibited interesting inhibition action to control proliferation of Trypanosoma cruzi, the parasite responsible for Chagas' disease. Some of these drugs were shown to be potent growth inhibitors of this parasite. All of these drugs had previously presented juvenoid activity on several non- related bug species such as Tenebrio molitor, Galleria mellonella, Dysdercus cingulatos, and Pyrrhocoris apterus.
Registro:
| Documento: | Artículo |
| Título: | Growth inhibitory effect of juvenile hormone analogues on epimastigotes of Trypanosoma cruzi |
| Autor: | Rodriguez, J.B.; Zhong, L.; Docampo, R.; Wimmer, Z.; Gros, E.G. |
| Filiación: | Depto. de Quimica Orgánica, Fac. de Cie. Exactas y Naturales, Universidad de Buenos Aires, 1428 Buenos Aires, Argentina Lab. of Molecular Parasitology, Department of Pathobiology, Univ. of Illinois at Urbana-C., 2001 South Lincoln Avenue, Urbana, IL 61801, United States Inst. for Organ. Chem./Biochem., Acad. of Sci. of the Czech Republic, Flemingovo námêsti 2, 16610 Prague 6, Czech Republic |
| Palabras clave: | benznidazole; fenoxycarb; hormone analog; ketoconazole; nifurtimox; article; drug mechanism; drug structure; epimastigote; growth inhibition; nonhuman; structure activity relation; Trypanosoma cruzi; Dysdercus; Galleria mellonella; Insecta; Pyrrhocoris apterus; Tenebrio molitor; Trypanosoma; Trypanosoma cruzi |
| Año: | 1998 |
| Volumen: | 8 |
| Número: | 22 |
| Página de inicio: | 3257 |
| Página de fin: | 3260 |
| DOI: | http://dx.doi.org/10.1016/S0960-894X(98)00590-3 |
| Título revista: | Bioorganic and Medicinal Chemistry Letters |
| Título revista abreviado: | Bioorg. Med. Chem. Lett. |
| ISSN: | 0960894X |
| CODEN: | BMCLE |
| CAS: | benznidazole, 22994-85-0; fenoxycarb, 72490-01-8; ketoconazole, 65277-42-1; nifurtimox, 23256-30-6 |
| Registro: | https://bibliotecadigital.exactas.uba.ar/collection/paper/document/paper_0960894X_v8_n22_p3257_Rodriguez |
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Citas:
---------- APA ----------
Rodriguez, J.B., Zhong, L., Docampo, R., Wimmer, Z. & Gros, E.G. (1998) . Growth inhibitory effect of juvenile hormone analogues on epimastigotes of Trypanosoma cruzi. Bioorganic and Medicinal Chemistry Letters, 8(22), 3257-3260.http://dx.doi.org/10.1016/S0960-894X(98)00590-3
---------- CHICAGO ----------
Rodriguez, J.B., Zhong, L., Docampo, R., Wimmer, Z., Gros, E.G. "Growth inhibitory effect of juvenile hormone analogues on epimastigotes of Trypanosoma cruzi" . Bioorganic and Medicinal Chemistry Letters 8, no. 22 (1998) : 3257-3260.http://dx.doi.org/10.1016/S0960-894X(98)00590-3
---------- MLA ----------
Rodriguez, J.B., Zhong, L., Docampo, R., Wimmer, Z., Gros, E.G. "Growth inhibitory effect of juvenile hormone analogues on epimastigotes of Trypanosoma cruzi" . Bioorganic and Medicinal Chemistry Letters, vol. 8, no. 22, 1998, pp. 3257-3260.http://dx.doi.org/10.1016/S0960-894X(98)00590-3
---------- VANCOUVER ----------
Rodriguez, J.B., Zhong, L., Docampo, R., Wimmer, Z., Gros, E.G. Growth inhibitory effect of juvenile hormone analogues on epimastigotes of Trypanosoma cruzi. Bioorg. Med. Chem. Lett. 1998;8(22):3257-3260.http://dx.doi.org/10.1016/S0960-894X(98)00590-3
