Artículo
Barolli, M.G.; Pomilio, A.B. "Synthesis of [131-I]-iodinated quercetin" (1997) Journal of Labelled Compounds and Radiopharmaceuticals. 39(11):927-933
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Abstract:
Two iodination procedures via thallation were applied to quercetin leading to the formation of 2'-iodoquercetin and 2',6,8-triiodoquercetin; their structures being elucidated by FT-IR and NMR spectral analysis. The preparation of mono- and polyiodinated products is discussed here on the basis of the experimental details and spectral data. This is the first report on the radiolabelling of quercetin, which is here selectively performed with 131-iodine. The radiochemical purity was of 99%.
Registro:
| Documento: | Artículo |
| Título: | Synthesis of [131-I]-iodinated quercetin |
| Autor: | Barolli, M.G.; Pomilio, A.B. |
| Filiación: | Depto. de Quim. Orgánica, Fac. de Ciencias Exactas y Naturales, Universidad de Buenos Aires, 1428 Buenos Aires, Argentina |
| Palabras clave: | 131-iodine; 2',6,8- triiodoquercetin; 2'-iodoquercetin; Iodination; Quercetin; Radiolabelling; iodine 131; quercetin; antioxidant activity; article; drug structure; drug synthesis; iodination; oxidative stress |
| Año: | 1997 |
| Volumen: | 39 |
| Número: | 11 |
| Página de inicio: | 927 |
| Página de fin: | 933 |
| DOI: | http://dx.doi.org/10.1002/(SICI)1099-1344(199711)39:11<927::AID-JLCR36>3.0.CO;2-6 |
| Título revista: | Journal of Labelled Compounds and Radiopharmaceuticals |
| Título revista abreviado: | J. LABEL. COMPD. RADIOPHARM. |
| ISSN: | 03624803 |
| CODEN: | JLCRD |
| CAS: | iodine 131, 10043-66-0, 15124-39-7; quercetin, 117-39-5 |
| Registro: | https://bibliotecadigital.exactas.uba.ar/collection/paper/document/paper_03624803_v39_n11_p927_Barolli |
Referencias:
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Citas:
---------- APA ----------
Barolli, M.G. & Pomilio, A.B. (1997) . Synthesis of [131-I]-iodinated quercetin. Journal of Labelled Compounds and Radiopharmaceuticals, 39(11), 927-933.http://dx.doi.org/10.1002/(SICI)1099-1344(199711)39:11<927::AID-JLCR36>3.0.CO;2-6
---------- CHICAGO ----------
Barolli, M.G., Pomilio, A.B. "Synthesis of [131-I]-iodinated quercetin" . Journal of Labelled Compounds and Radiopharmaceuticals 39, no. 11 (1997) : 927-933.http://dx.doi.org/10.1002/(SICI)1099-1344(199711)39:11<927::AID-JLCR36>3.0.CO;2-6
---------- MLA ----------
Barolli, M.G., Pomilio, A.B. "Synthesis of [131-I]-iodinated quercetin" . Journal of Labelled Compounds and Radiopharmaceuticals, vol. 39, no. 11, 1997, pp. 927-933.http://dx.doi.org/10.1002/(SICI)1099-1344(199711)39:11<927::AID-JLCR36>3.0.CO;2-6
---------- VANCOUVER ----------
Barolli, M.G., Pomilio, A.B. Synthesis of [131-I]-iodinated quercetin. J. LABEL. COMPD. RADIOPHARM. 1997;39(11):927-933.http://dx.doi.org/10.1002/(SICI)1099-1344(199711)39:11<927::AID-JLCR36>3.0.CO;2-6
