Artículo

Vitale, A.A.; Calvino, M.A.; Ferrari, C.C.; Stahl, A.E.; Pomilio, A.B. "Preparation and biological evaluation of technetium‐99m‐phenylethylamine complexes" (1995) Journal of Labelled Compounds and Radiopharmaceuticals. 36(6):509-519
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Abstract:

Biological and chemical characteristics of 99mTc‐phenethylamines complexes are presented. 2‐(4,5‐Dimethoxy‐2‐nitrophenyl)ethylamine, 2‐(3,4‐dimethoxyphenyl)ethylamine and 2‐(2‐amino‐4,5‐dimethoxyphenyl)‐ethylamine were used as ligands. A preliminary evaluation of these 99mTc‐complexes as dopamine receptor radioligands was also performed. Net charges at each atom were also calculated by a semiempirical ZINDO/1 method for comparison of free ligands' parameters with those of the respective technetium‐complexes. Copyright © 1995 John Wiley & Sons, Ltd.

Registro:

Documento: Artículo
Título:Preparation and biological evaluation of technetium‐99m‐phenylethylamine complexes
Autor:Vitale, A.A.; Calvino, M.A.; Ferrari, C.C.; Stahl, A.E.; Pomilio, A.B.
Filiación:CONICET, Departamento de Química Orgánica, Facultad de Ciencias Exactas y Naturales, Universidad de Buenos Aires, Ciudad Universitaria, Pabellón 2, Buenos Aires, 1428, Argentina
Ineuci-Conicet, Departamento de Ciencias Biológicas, Fcen, Uba, Argentina
Palabras clave:2‐(2‐Amino‐4,5‐dimethoxyphenyl)ethylamine; 2‐(3,4‐Dimethoxyphenyl)‐ethylamine; 2‐(4,5‐Dimethoxy‐2‐nitrophenyl)ethylamine; 99m‐Technetium complexes; Biodistribution; Preparation; semiempirical ZINDO/1 calculations; phenethylamine derivative; technetium 99m; technetium complex; animal experiment; article; brain; controlled study; drug distribution; drug structure; drug synthesis; electrophoresis; female; intracerebral drug administration; isotope labeling; nonhuman; radiochromatography; rat; Animalia
Año:1995
Volumen:36
Número:6
Página de inicio:509
Página de fin:519
DOI: http://dx.doi.org/10.1002/jlcr.2580360602
Título revista:Journal of Labelled Compounds and Radiopharmaceuticals
Título revista abreviado:J. Label. Compd. Radiopharm.
ISSN:03624803
Registro:https://bibliotecadigital.exactas.uba.ar/collection/paper/document/paper_03624803_v36_n6_p509_Vitale

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Citas:

---------- APA ----------
Vitale, A.A., Calvino, M.A., Ferrari, C.C., Stahl, A.E. & Pomilio, A.B. (1995) . Preparation and biological evaluation of technetium‐99m‐phenylethylamine complexes. Journal of Labelled Compounds and Radiopharmaceuticals, 36(6), 509-519.
http://dx.doi.org/10.1002/jlcr.2580360602
---------- CHICAGO ----------
Vitale, A.A., Calvino, M.A., Ferrari, C.C., Stahl, A.E., Pomilio, A.B. "Preparation and biological evaluation of technetium‐99m‐phenylethylamine complexes" . Journal of Labelled Compounds and Radiopharmaceuticals 36, no. 6 (1995) : 509-519.
http://dx.doi.org/10.1002/jlcr.2580360602
---------- MLA ----------
Vitale, A.A., Calvino, M.A., Ferrari, C.C., Stahl, A.E., Pomilio, A.B. "Preparation and biological evaluation of technetium‐99m‐phenylethylamine complexes" . Journal of Labelled Compounds and Radiopharmaceuticals, vol. 36, no. 6, 1995, pp. 509-519.
http://dx.doi.org/10.1002/jlcr.2580360602
---------- VANCOUVER ----------
Vitale, A.A., Calvino, M.A., Ferrari, C.C., Stahl, A.E., Pomilio, A.B. Preparation and biological evaluation of technetium‐99m‐phenylethylamine complexes. J. Label. Compd. Radiopharm. 1995;36(6):509-519.
http://dx.doi.org/10.1002/jlcr.2580360602