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Abstract:

The influence of methoxamine on the contractile tension of isolated rat abdominal aorta, and on its capacity to produce a platelet antiaggregating substance, were explored. Methoxamine stimulated platelet antiaggregation and diminished arterial tone. The last action was blocked by phentolamine as well as by inhibitiors of cyclo-oxygenase and prostacyclinsynthetase. © 1983 Birkhäuser Verlag.

Registro:

Documento: Artículo
Título:Is prostacyclin subserving a vasodilator effect of methoxamine involving alpha adrenoreceptors?
Autor:Borda, E.; Sterin-Borda, L.; Gimeno, M.F.; Lazzari, M.; Gimeno, A.L.
Filiación:Centro de Estudios Farmacológicos y de Principios Naturales (CEFAPRIN), Consejo Nacional de Investigaciones Cientificas y Técnicas, de la República Argentina (CONICET), Serrano 665/69, Buenos Aires, 1414, Argentina
Instituto de Investigaciones Hematológicas, Academia Nacional de Medicina, Serrano 665/69, Buenos Aires, 1414, Argentina
Palabras clave:4 aminophenol; acetylsalicylic acid; alpha adrenergic receptor; indometacin; methoxamine; phentolamine; propranolol; prostacyclin; prostacyclin synthase; tranylcypromine; animal cell; ant; aorta; drug efficacy; great blood vessel; nonhuman; rat; Animals; Aorta, Abdominal; Epoprostenol; Indomethacin; Male; Methoxamine; Muscle Contraction; Platelet Aggregation; Prostaglandins; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Vasodilator Agents; Animalia; Formicidae
Año:1983
Volumen:39
Número:8
Página de inicio:894
Página de fin:896
DOI: http://dx.doi.org/10.1007/BF01990425
Título revista:Experientia
Título revista abreviado:Experientia
ISSN:00144754
CODEN:EXPEA
CAS:4 aminophenol, 123-30-8; acetylsalicylic acid, 493-53-8, 50-78-2, 53663-74-4, 53664-49-6, 63781-77-1; indometacin, 53-86-1, 74252-25-8, 7681-54-1; methoxamine, 390-28-3, 61-16-5; phentolamine, 50-60-2, 73-05-2; propranolol, 13013-17-7, 318-98-9, 3506-09-0, 4199-09-1, 525-66-6; prostacyclin, 35121-78-9, 61849-14-7; prostacyclin synthase, 65802-86-0; tranylcypromine, 13492-01-8, 155-09-9, 54-97-7; Epoprostenol, 35121-78-9; Indomethacin, 53-86-1; Methoxamine, 390-28-3; Prostaglandins; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Vasodilator Agents
Registro:https://bibliotecadigital.exactas.uba.ar/collection/paper/document/paper_00144754_v39_n8_p894_Borda

Referencias:

  • Wesffall, T.C., (1977) Physiol. Rev., 57, p. 659
  • Baumann, J., Bruchhausen, F., Wurm, G., (1979) Naunyn Schmiedeberg's Arch. Pharmak., 307, p. 73
  • Flower, R.J., Blackwell, G.I., (1976) Biochem. Pharmac., 25, p. 285
  • Borda, E.S., del Agostini, M.C., Gimeno, M.F., Gimeno, A.L., (1981) Pharmac. Res. Commun., 13, p. 981
  • Borda, E.S., del Agostini, M.C., Sterin-Speziale, N., Gimeno, M.F., Gimeno, A.L., (1979) Prostaglandins, 18, p. 829
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  • Borda, L., Schuchleih, R., Henry, P., (1980) Circulation Res., 46, p. 878
  • Borda, E.S., Sauvage, J., Sterin-Borda, L., Gimeno, M.F., Gimeno, A.L., (1979) Eur. J. Pharmac., 56, p. 61
  • Borda, E.S., del Agostini, M.C., Gimeno, M.F., Gimeno, A.L., (1981) Pharmac. Res. Commun., 13, p. 487
  • Vane, J.R., (1971) Nature New Biol., 231, p. 232
  • Moncada, S., (1982) Br. J. Pharmac., 76, p. 3
  • Sterin-Borda, L., Borda, E.S., Gimeno, M.F., Lazzari, M.L., del Castillo, E., Gimeno, A.L., (1982) Diabetologia, 22, p. 56
  • Gryglewsky, R.J., Bunting, S., Flower, R., Vane, J.R., (1976) Prostaglandins, 12, p. 685
  • Brückner-Schmidt, R., Jackisch, R., Hertting, G., (1981) Naunyn Schmiedeberg's Arch. Pharmak., 316, p. 1

Citas:

---------- APA ----------
Borda, E., Sterin-Borda, L., Gimeno, M.F., Lazzari, M. & Gimeno, A.L. (1983) . Is prostacyclin subserving a vasodilator effect of methoxamine involving alpha adrenoreceptors?. Experientia, 39(8), 894-896.
http://dx.doi.org/10.1007/BF01990425
---------- CHICAGO ----------
Borda, E., Sterin-Borda, L., Gimeno, M.F., Lazzari, M., Gimeno, A.L. "Is prostacyclin subserving a vasodilator effect of methoxamine involving alpha adrenoreceptors?" . Experientia 39, no. 8 (1983) : 894-896.
http://dx.doi.org/10.1007/BF01990425
---------- MLA ----------
Borda, E., Sterin-Borda, L., Gimeno, M.F., Lazzari, M., Gimeno, A.L. "Is prostacyclin subserving a vasodilator effect of methoxamine involving alpha adrenoreceptors?" . Experientia, vol. 39, no. 8, 1983, pp. 894-896.
http://dx.doi.org/10.1007/BF01990425
---------- VANCOUVER ----------
Borda, E., Sterin-Borda, L., Gimeno, M.F., Lazzari, M., Gimeno, A.L. Is prostacyclin subserving a vasodilator effect of methoxamine involving alpha adrenoreceptors?. Experientia. 1983;39(8):894-896.
http://dx.doi.org/10.1007/BF01990425